SCHEMBL9728830

SCHEMBL9728830

O=C(Nc1nc(=O)[nH]c2ccccc12)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 9/20 0.58
APP P05067 2/20 0.56
ABCG2 Q9UNQ0 1/20 0.54
MAOB P27338 2/20 0.51
ADORA2A P29274 2/20 0.51
NPC1 O15118 1/20 0.51
PKM P14618 1/20 0.51
RAB9A P51151 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
BRD4 O60885 1/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
TSHR P16473 1/20 0.49
HSD17B10 Q99714 1/20 0.49
PARP14 Q460N5 1/20 0.48
LMNA P02545 1/20 0.48
SCD O00767 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3344881 0.78 APP (0.54) ADORA3APPSMN1; SMN2KDM4EALDH1A1
SCHEMBL627899 0.77 FGFR1 (0.65)
SCHEMBL31040239 0.77 FGFR1 (0.65)
SCHEMBL9728941 0.77 NPC1 (0.67) MAOBADORA2ANPC1PKMRAB9A
SCHEMBL20427956 0.77 LMNA (0.48) ADORA3ABCG2MAOBADORA2ANPC1
SCHEMBL31347645 0.75 APP (0.61) ADORA3APPABCG2KDM4EALDH1A1
SCHEMBL2395706 0.75 APP (0.61) ADORA3APPABCG2KDM4EALDH1A1
SCHEMBL29044810 0.74 APP (0.60) ADORA3APPSMN1; SMN2KDM4EALDH1A1
SCHEMBL29033598 0.74 ADORA3 (0.62) ADORA3APPKDM4EALDH1A1HPGD
SCHEMBL31060760 0.73 ADORA3 (1.00) ADORA3NPC1RAB9ASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084457-A Cognition activators and nervous system disorders AMERICAN CYANAMID COMPANY (US) 1992-01-28 US disclosed
US-5001157-A Substituted N-[[2-(aminocarbonyl)phenylamino]thioxomethyl]benzamides AMERICAN CYANAMID COMPANY (US) 1991-03-19 US disclosed