SCHEMBL9729382

SCHEMBL9729382

O=C1CCC(c2cccc(Cl)c2)(c2cccc(Cl)c2)C2CN(Cc3ccccc3)CC12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.46
CXCR3 P49682 4/20 0.46
SIGMAR1 Q99720 2/20 0.42
CHRM2 P08172 1/20 0.41
CHRM3 P20309 1/20 0.41
CCR5 P51681 1/20 0.41
MAPT P10636 2/20 0.41
TACR1 P25103 2/20 0.41
MEN1 O00255 1/20 0.41
CYP3A4 P08684 1/20 0.41
TSHR P16473 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
DOCK5 Q9H7D0 1/20 0.40
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9003055 0.90 TACR1 (0.48) CXCR3MAPTTACR1MEN1CYP3A4
SCHEMBL9003052 0.90 TACR1 (0.48) CXCR3MAPTTACR1MEN1CYP3A4
SCHEMBL9268452 0.90 TACR1 (0.48) CXCR3MAPTTACR1MEN1CYP3A4
SCHEMBL9729281 0.88 MEN1 (0.43) DPP4CXCR3SIGMAR1CHRM2CHRM3
SCHEMBL9729536 0.88 CCR5 (0.42) DPP4CXCR3SIGMAR1CHRM2CHRM3
SCHEMBL9729490 0.82 TACR1 (0.48) MAPTTACR1MEN1CYP3A4TSHR
SCHEMBL8874365 0.80 GAA (0.44) DPP4MAPTTACR1MEN1CYP3A4
SCHEMBL9730167 0.78 MEN1 (0.51) SIGMAR1CHRM2CHRM3CCR5MAPT
SCHEMBL9729134 0.77 TACR1 (0.39) DPP4CXCR3SIGMAR1MAPTTACR1
SCHEMBL8875025 0.76 GAA (0.46) DPP4TACR1DRD2DRD3GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112988-A ISOINDOLONE DERIVATIVES RHONE-POULENC SANTE (FR) 1992-05-12 US disclosed
US-5102667-A Antiallergens, antiinflammatory agents, nervous system disorders, immunology, psychological disorders RHONE-POULENC SANTE (FR) 1992-04-07 US disclosed