SCHEMBL9729134

SCHEMBL9729134

O=C1CCC(c2ccccc2F)(c2ccccc2F)C2CN(Cc3ccccc3)CC12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 5/20 0.39
SCN5A Q14524 1/20 0.37
SCN9A Q15858 1/20 0.37
CXCR3 P49682 2/20 0.37
SIGMAR1 Q99720 3/20 0.37
CYP3A4 P08684 2/20 0.36
TSHR P16473 2/20 0.36
CYP2C19 P33261 2/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
FUCA1 P04066 2/20 0.36
DPP4 P27487 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9003052 0.84 TACR1 (0.48) TACR1CXCR3CYP3A4TSHRCYP2C19
SCHEMBL9268452 0.84 TACR1 (0.48) TACR1CXCR3CYP3A4TSHRCYP2C19
SCHEMBL9003055 0.84 TACR1 (0.48) TACR1CXCR3CYP3A4TSHRCYP2C19
SCHEMBL9729536 0.81 CCR5 (0.42) TACR1CXCR3SIGMAR1CYP3A4TSHR
SCHEMBL8875025 0.78 GAA (0.46) TACR1DRD2DRD3FUCA1DPP4
SCHEMBL9729382 0.77 DPP4 (0.46) TACR1CXCR3SIGMAR1CYP3A4TSHR
SCHEMBL8874365 0.77 GAA (0.44) TACR1CYP3A4TSHRCYP2C19ALDH1A1
SCHEMBL9729281 0.76 MEN1 (0.43) TACR1CXCR3SIGMAR1CYP3A4TSHR
SCHEMBL8874334 0.75 TACR1 (0.40) TACR1SIGMAR1CYP3A4TSHRCYP2C19
SCHEMBL8875253 0.73 CHRM4 (0.44) TACR1SCN9ASIGMAR1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112988-A ISOINDOLONE DERIVATIVES RHONE-POULENC SANTE (FR) 1992-05-12 US disclosed
US-5102667-A Antiallergens, antiinflammatory agents, nervous system disorders, immunology, psychological disorders RHONE-POULENC SANTE (FR) 1992-04-07 US disclosed