SCHEMBL9729781

SCHEMBL9729781

CCOC(=O)c1cc(Cl)c2cc(C)ccc2n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
KDM4E B2RXH2 4/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
MAPK1 P28482 2/20 0.53
TDP1 Q9NUW8 1/20 0.53
LMNA P02545 1/20 0.53
CYP1A2 P05177 1/20 0.46
MAPT P10636 3/20 0.46
HPGD P15428 2/20 0.45
GLA P06280 1/20 0.45
POLB P06746 1/20 0.45
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45
GABRA2 P47869 1/20 0.45
GABRB2 P47870 1/20 0.45
PKM P14618 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2652933 0.85 CTSL (0.61) ALDH1A1SMN1; SMN2KDM4ETDP1LMNA
SCHEMBL163381 0.84 SMN1; SMN2 (0.53) ALDH1A1SMN1; SMN2KDM4ETDP1LMNA
SCHEMBL3350745 0.82 LMNA (0.62) ALDH1A1KDM4EL3MBTL1LMNAMAPT
SCHEMBL23198535 0.81 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2KDM4EL3MBTL1CYP1A2
SCHEMBL28883896 0.81 KDM4E (0.54) ALDH1A1SMN1; SMN2KDM4EL3MBTL1MAPK1
SCHEMBL31254231 0.81 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2KDM4EL3MBTL1CYP1A2
SCHEMBL22292210 0.80 KDM4E (0.62) ALDH1A1SMN1; SMN2KDM4EL3MBTL1MAPK1
SCHEMBL9724191 0.80 LMNA (0.58) SMN1; SMN2LMNAPKM
SCHEMBL20944487 0.80 MEN1 (0.60) ALDH1A1L3MBTL1LMNAMAPTHPGD
SCHEMBL9319008 0.80 TNF (0.50) ALDH1A1SMN1; SMN2KDM4ELMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112837-A Inhibitors of thymidylate synthetase enzyme IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-05-12 US disclosed
EP-0318225-A2 6-Aryl aminomethyl quinoline derivatives and their use as anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-31 EP disclosed