SCHEMBL9730918

SCHEMBL9730918

CC(C)c1nnn(-c2ccc(F)cc2)c1CCl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.39
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
SLC5A1 P13866 1/20 0.37
SLC5A2 P31639 1/20 0.37
GABRA5 P31644 3/20 0.36
GABRG2 P18507 2/20 0.36
GABRB3 P28472 2/20 0.36
KCNH2 Q12809 1/20 0.36
PPARA Q07869 1/20 0.36
LMNA P02545 3/20 0.36
ALDH1A1 P00352 3/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.34
MAPT P10636 3/20 0.34
NPC1 O15118 2/20 0.34
TSHR P16473 1/20 0.34
RAB9A P51151 1/20 0.34
DCTPP1 Q9H773 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9730089 0.85 ALDH1A1 (0.43) PTGS2IDO1TDO2SLC5A1SLC5A2
SCHEMBL9730309 0.80 PTGS2 (0.45) PTGS2IDO1TDO2GABRA5GABRG2
Hydrochloric Acid SCHEMBL9730988 0.77 IDO1 (0.38) PTGS2IDO1TDO2SLC5A1SLC5A2
SCHEMBL9730226 0.74 PTGS2 (0.43) PTGS2IDO1TDO2SLC5A1SLC5A2
SCHEMBL498069 0.73 NR1H4 (0.45) GABRB3
SCHEMBL9730322 0.71 HMGCR (0.50)
SCHEMBL17699229 0.71 ALDH1A1 (0.44) PTGS2IDO1TDO2SLC5A1SLC5A2
SCHEMBL21834124 0.70 GABRA5 (0.46) PTGS2IDO1TDO2GABRA5GABRG2
SCHEMBL2683661 0.67 PTGS2 (0.49) PTGS2SLC5A1SLC5A2GABRA5GABRG2
Hydrochloric Acid SCHEMBL10533684 0.66 KDM4E (0.40) LMNAALDH1A1L3MBTL1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5081136-A 1,2,3-TRIAZOLE COMPOUNDS ACTIVE AS INHIBITORS OF THE ENZYME HMG-COA REDUCTASE AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ZAMBON GROUP S.P.A. (IT) 1992-01-14 US disclosed
EP-0433842-A2 1,2,3-Triazole derivatives active as inhibitors of the enzyme HMG-COA reductase and pharmaceutical compositions containing them ZAMBON GROUP S.p.A. (IT) 1991-06-26 EP disclosed