SCHEMBL9733117

SCHEMBL9733117

COc1cccc(Cn2cc(C=O)c3ccccc32)c1

nearest known ligand 0.73

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.67
SMN1; SMN2 Q16637 7/20 0.67
LMNA P02545 5/20 0.67
TDP1 Q9NUW8 2/20 0.67
KMT2A Q03164 3/20 0.65
MEN1 O00255 2/20 0.65
POLB P06746 2/20 0.60
L3MBTL1 Q9Y468 1/20 0.58
HTT P42858 3/20 0.57
ABCC2 Q92887 1/20 0.57
MAPT P10636 5/20 0.56
NPSR1 Q6W5P4 1/20 0.56
BCHE P06276 1/20 0.53
NPC1 O15118 1/20 0.52
HPGD P15428 1/20 0.52
RAB9A P51151 1/20 0.52
TP53 P04637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28239560 0.90 POLB (0.60) ALDH1A1SMN1; SMN2LMNATDP1KMT2A
SCHEMBL797463 0.86 ALDH1A1 (0.69) ALDH1A1SMN1; SMN2LMNATDP1KMT2A
SCHEMBL9733878 0.85 ALDH1A1 (0.65) ALDH1A1SMN1; SMN2LMNATDP1KMT2A
SCHEMBL8685723 0.85 SLC2A1 (0.55) ALDH1A1SMN1; SMN2LMNATDP1KMT2A
SCHEMBL28900440 0.84 ALDH1A1 (0.75) ALDH1A1SMN1; SMN2LMNATDP1KMT2A
SCHEMBL9584018 0.84 PLA2G2A (0.61) ALDH1A1LMNABCHE
SCHEMBL13131367 0.82 MAPT (0.57) ALDH1A1LMNAKMT2APOLBABCC2
SCHEMBL18509023 0.82 MAPT (0.56) LMNAKMT2AMEN1POLBABCC2
SCHEMBL28530692 0.81 ABCC2 (0.60) ALDH1A1SMN1; SMN2LMNATDP1KMT2A
SCHEMBL28477087 0.81 BCHE (0.55) ALDH1A1SMN1; SMN2LMNATDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108358923-B Sophoridine pyrrole and indole derivatives, and preparation method and application thereof 广西大学 2020-11-03 CN claimed
CN-108047226-B Matrine pyrrole and indole derivatives, and preparation method and application thereof 广西大学 2020-11-03 CN claimed
CN-108358923-A Sophoridine pyrroles, indole derivatives and the preparation method and application thereof 广西大学 2018-08-03 CN claimed
WO-1992007829-A1 INDOLE-3-METHANAMINES USEFUL AS ANTI-DIABETIC, ANTI-OBESITY AND ANTI-ATHEROSCLEROTIC AGENTS THE UPJOHN COMPANY (US) 1992-05-14 WO disclosed