SCHEMBL9733548

SCHEMBL9733548

COc1cc(CN2CCCN(Cc3cc(OC)cc(OC)c3O)C2)c(O)c(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.50
KDM4E B2RXH2 4/20 0.50
MAPT P10636 4/20 0.46
MAPK1 P28482 2/20 0.46
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
LMNA P02545 1/20 0.43
HTR1A P08908 1/20 0.43
ADRA2A P08913 1/20 0.43
CYP2D6 P10635 1/20 0.43
ADRA2C P18825 1/20 0.43
OPRK1 P41145 1/20 0.43
KCNH2 Q12809 1/20 0.43
EBP Q15125 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
MPO P05164 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9734968 0.87 GAA (0.51) GAAKDM4EMAPTMAPK1LMNA
SCHEMBL9733677 0.82 CA1 (0.53) GAAKDM4EMAPTMAPK1TDP1
SCHEMBL9733717 0.79 GAA (0.50) GAAKDM4EMEN1KMT2A
SCHEMBL9734162 0.78 GAA (0.79) GAAKDM4EMAPTMAPK1TDP1
SCHEMBL9734550 0.76 KDM4E (0.53) GAAKDM4ETDP1L3MBTL1MPO
SCHEMBL9734499 0.76 GAA (0.69) GAAKDM4EMAPTMAPK1TDP1
SCHEMBL29274523 0.73 GAA (0.66) GAAKDM4ETDP1L3MBTL1MEN1
SCHEMBL29274529 0.72 GAA (0.68) GAAKDM4EMAPTMAPK1TDP1
SCHEMBL3833937 0.72 PDE4A (0.48) MAPK1
SCHEMBL3100738 0.71 GAA (0.56) GAAKDM4EMAPTMAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5106975-A Hexahydropyrimidine derivatives ETHYL PETROLEUM ADDITIVES, INC. (US) 1992-04-21 US disclosed