SCHEMBL9733717

SCHEMBL9733717

C=CCc1cc(CN2CCCN(Cc3cc(CC=C)cc(OC)c3O)C2)c(O)c(OC)c1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.50
TNKS O95271 1/20 0.50
TNKS2 Q9H2K2 1/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 3/20 0.45
CYP3A4 P08684 2/20 0.45
ALOX5 P09917 1/20 0.45
AR P10275 1/20 0.45
PTGS1 P23219 1/20 0.45
TRPM8 Q7Z2W7 1/20 0.45
TSHR P16473 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
CCR3 P51677 1/20 0.43
PPARG P37231 1/20 0.41
PPARD Q03181 1/20 0.41
PPARA Q07869 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733617 0.89 ALDH1A1 (0.49) GAATNKSTNKS2KDM4EALDH1A1
SCHEMBL13899835 0.81 TNKS (0.63) GAATNKSTNKS2KDM4EALDH1A1
SCHEMBL31255953 0.81 TNKS (0.63) GAATNKSTNKS2KDM4EALDH1A1
SCHEMBL9734968 0.80 GAA (0.51) GAAKDM4EALOX5MEN1KMT2A
SCHEMBL17649934 0.80 KDM4E (0.51) GAATNKSTNKS2KDM4EALDH1A1
SCHEMBL6554990 0.79 TNKS (0.65) TNKSTNKS2ALDH1A1CYP3A4ALOX5
SCHEMBL9733548 0.79 GAA (0.50) GAAKDM4EMEN1KMT2A
SCHEMBL9734162 0.78 GAA (0.79) GAAKDM4EALDH1A1SMN1; SMN2
SCHEMBL1005864 0.77 TNKS (0.61) GAATNKSTNKS2KDM4EALDH1A1
SCHEMBL29274523 0.76 GAA (0.66) GAAKDM4EALDH1A1TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5106975-A Hexahydropyrimidine derivatives ETHYL PETROLEUM ADDITIVES, INC. (US) 1992-04-21 US disclosed
EP-0434185-A2 Hexahydropyrimidine derivatives ETHYL PETROLEUM ADDITIVES, INC. (US) 1991-06-26 EP disclosed