SCHEMBL9733795

SCHEMBL9733795

CC1(C)Cc2ccc(Br)cc2C2OC21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
HTR2B P41595 1/20 0.36
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
ALDH1A1 P00352 2/20 0.32
POLB P06746 1/20 0.32
TSHR P16473 1/20 0.32
ADRA2A P08913 2/20 0.32
PNMT P11086 2/20 0.32
ADRA2B P18089 2/20 0.32
ADRA2C P18825 2/20 0.32
PDE4B Q07343 1/20 0.32
LMNA P02545 1/20 0.31
MAPK1 P28482 1/20 0.31
KDM1A O60341 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
DRD2 P14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733609 0.78 SIGMAR1 (0.38) HTR2AALDH1A1TSHRADRA2AADRA2B
SCHEMBL9733546 0.77 ABCB1 (0.41) LMNAKDM1ADRD2
SCHEMBL9240188 0.75 KDM1A (0.40) HTR2AHTR2CHTR2BOPRM1OPRD1
SCHEMBL29804038 0.75 KDM1A (0.40) HTR2AHTR2CHTR2BOPRM1OPRD1
SCHEMBL29122626 0.75 HTR2A (0.39) HTR2AHTR2CHTR2BOPRM1OPRD1
SCHEMBL27795745 0.71 HTR2A (0.36) HTR2AHTR2CHTR2BOPRM1OPRD1
SCHEMBL9141916 0.69 HTR2A (0.36) HTR2AHTR2CHTR2BADRA2AADRA2C
SCHEMBL9733411 0.68 OPRM1 (0.38) HTR2AHTR2CHTR2BOPRM1OPRD1
SCHEMBL23361915 0.67 CNR2 (0.41) HTR2AHTR2CHTR2BOPRM1OPRD1
SCHEMBL9141090 0.67 MEN1 (0.43) HTR2AHTR2CHTR2BOPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed