SCHEMBL9733860

SCHEMBL9733860

COC(=O)C(C)C(=O)Cc1ccc(SC(=O)N(C)C)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
ACHE P22303 2/20 0.34
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
PTPRB P23467 1/20 0.32
GAA P10253 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
HTT P42858 1/20 0.32
CYP4F2 P78329 1/20 0.32
CYP4A11 Q02928 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
CA12 O43570 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32
MAPT P10636 1/20 0.32
TSHR P16473 1/20 0.32
BMP1 P13497 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9780186 0.81 SLC6A4 (0.46) ALDH1A1MAPTTSHR
SCHEMBL377862 0.80 CYP4F2 (0.51) ALDH1A1GAACYP4F2CYP4A11MAPT
SCHEMBL9780325 0.77 ALDH1A1 (0.38) ALDH1A1GAATAS1R3TAS1R1MAPT
SCHEMBL9734555 0.76 ESR1 (0.53) GAAESR1ESR2HTTMAPT
SCHEMBL9733733 0.75 HTT (0.57) ALDH1A1HTTPOLB
SCHEMBL9780185 0.75 HTT (0.38) ALDH1A1PTPRBGAAESR1ESR2
SCHEMBL6541372 0.75 CA2 (0.47) ALDH1A1GAAHTTMAPTTSHR
SCHEMBL10911841 0.73 L3MBTL1 (0.36) ALDH1A1PTPRBGAAESR1ESR2
SCHEMBL4676623 0.72 PPARG (0.43) PPARGPPARAMAPTPOLBMEN1
SCHEMBL20244667 0.72 ALDH1A1 (0.53) ALDH1A1ACHEHTTMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135940-A Antiallegens, antiinflammatory agents MERCK FROSST CANADA, INC. (CA) 1992-08-04 US disclosed
EP-0252639-A1 Leukotriene antagonists MERCK FROSST CANADA INC. (CA) 1988-01-13 EP disclosed
EP-0104885-B1 LEUKOTRIENE ANTAGONISTS, THEIR PRODUCTION, AND COMPOSITIONS CONTAINING THEM MERCK FROSST CANADA INC. (CA) 1986-06-04 EP disclosed