SCHEMBL9734002

SCHEMBL9734002

NS(=O)(=O)c1cc2c(=O)n(-c3ccccc3Cl)c(CBr)nc2s1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 8/20 0.47
ALDH1A1 P00352 4/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C19 P33261 2/20 0.40
KDM4E B2RXH2 2/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
POLB P06746 1/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HSP90AA1 P07900 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733487 0.92 MALT1 (0.39) MALT1ALDH1A1CYP2D6CYP2C19KDM4E
SCHEMBL9733604 0.89 ALDH1A1 (0.41) MALT1ALDH1A1CYP2D6CYP2C19KDM4E
SCHEMBL9733681 0.89 ALDH1A1 (0.45) MALT1ALDH1A1CYP2D6CYP2C19KDM4E
SCHEMBL9733850 0.88 ALDH1A1 (0.41) MALT1ALDH1A1CYP2D6CYP2C19KDM4E
SCHEMBL9733299 0.88 ALDH1A1 (0.47) MALT1ALDH1A1CYP2D6CYP2C19KDM4E
SCHEMBL9733701 0.86 ALDH1A1 (0.47) MALT1ALDH1A1CYP2D6CYP2C19KDM4E
SCHEMBL9733424 0.84 ALDH1A1 (0.44) ALDH1A1CYP2D6CYP2C19KDM4ELMNA
SCHEMBL9734019 0.84 ALDH1A1 (0.59) ALDH1A1CYP2D6CYP2C19KDM4ELMNA
SCHEMBL9733685 0.83 CA2 (0.41) MALT1ALDH1A1CYP2D6CYP2C19KDM4E
SCHEMBL9734163 0.83 HIF1A (0.48) ALDH1A1CYP2D6CYP2C19HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5124331-A Anticancer agents YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1992-06-23 US disclosed
EP-0364598-A1 3,4-dihydrothieno ¬2,3-d pyrimidine compounds and pharmaceutical application thereof YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1990-04-25 EP disclosed