SCHEMBL9736896

SCHEMBL9736896

CCCCn1c(=O)[nH]c(=O)c2c(-c3ccc(F)cc3)c(C=CC=O)c(C(C)C)nc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.45
ALDH1A1 P00352 6/20 0.41
HTT P42858 3/20 0.40
MEN1 O00255 5/20 0.40
KMT2A Q03164 5/20 0.40
TDP1 Q9NUW8 1/20 0.38
MAPK1 P28482 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PDE4A P27815 1/20 0.36
ADORA2A P29274 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
GCGR P47871 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9388048 1.00 KDM4E (0.45) KDM4EALDH1A1HTTMEN1KMT2A
SCHEMBL9384186 0.91 GCGR (0.38) KDM4EALDH1A1MAPK1RXFP1PDE4A
SCHEMBL9383396 0.91 KDM4E (0.48) KDM4EALDH1A1HTTMEN1KMT2A
SCHEMBL9735137 0.91 GCGR (0.38) KDM4EALDH1A1MAPK1RXFP1PDE4A
SCHEMBL9736133 0.86 GCGR (0.37) ALDH1A1KMT2ACYP1A2CYP2C19SMN1; SMN2
SCHEMBL9736123 0.86 GCGR (0.37) ALDH1A1KMT2ACYP1A2CYP2C19SMN1; SMN2
SCHEMBL9734749 0.85 KDM4E (0.44) KDM4EALDH1A1HTTMAPK1RXFP1
SCHEMBL9734676 0.82 HMGCR (0.43) KDM4EALDH1A1HTTRXFP1CYP3A4
SCHEMBL9734698 0.82 HMGCR (0.43) KDM4EALDH1A1HTTRXFP1CYP3A4
SCHEMBL9387249 0.82 GCGR (0.54) KDM4EALDH1A1HTTGCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5145959-A Enzyme inhibitors; antilipemic agents; treatment of atherosclerosis BAYER AKTIENGESELLSCHAFT (DE) 1992-09-08 US disclosed
US-5075311-A Anticholesterol agents BAYER AKTIENGESELLSCHAFT (DE) 1991-12-24 US disclosed