SCHEMBL9523672

SCHEMBL9523672

CC(C)c1nc2[nH]c(=O)ccc2c(-c2ccc(F)cc2)c1/C=C/C=O

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GCGR P47871 6/20 0.40
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
ESR1 P03372 1/20 0.35
HMGCR P04035 1/20 0.35
CHRM1 P11229 1/20 0.35
TBXA2R P21731 1/20 0.35
PDE4A P27815 1/20 0.35
ADRA1A P35348 1/20 0.35
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
MAPK13 O15264 4/20 0.34
MAPK12 P53778 4/20 0.34
MAPK11 Q15759 4/20 0.34
MAPK14 Q16539 4/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9791356 1.00 GCGR (0.40) GCGRADORA2AADORA1ESR1HMGCR
SCHEMBL9524280 0.89 GCGR (0.43) GCGRADORA2AADORA1PDE3BPDE3A
SCHEMBL9727600 0.84 GCGR (0.41) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL9698874 0.84 GCGR (0.41) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL8949683 0.81 GCGR (0.53) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL9735571 0.80 GCGR (0.39) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL9383069 0.80 GCGR (0.39) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL8949786 0.78 GCGR (0.47) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL9791355 0.77 HMGCR (0.47) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL9380517 0.77 RXRA (0.47) GCGRESR1HMGCRCHRM1TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0391185-B1 Substituted 1,8-naphthyridines BAYER AG (DE) 1993-12-29 EP disclosed
US-5034399-A Enzyme inhibitors, anticholesterol agents or antilipemic agents BAYER AKTIENGESELLSCHAFT (DE) 1991-07-23 US disclosed
EP-0391185-A1 Substituted 1,8-naphthyridines BAYER AG (DE) 1990-10-10 EP disclosed