SCHEMBL9737111

SCHEMBL9737111

CC(Nc1cc(C(=O)O)cc(S(N)(=O)=O)c1Cl)c1cccc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 1/20 0.42
SCN5A Q14524 1/20 0.42
SCN8A Q9UQD0 1/20 0.42
CYP2D6 P10635 2/20 0.41
IDH1 O75874 1/20 0.40
CASR P41180 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
METAP2 P50579 1/20 0.39
METAP1 P53582 1/20 0.39
AURKA O14965 1/20 0.39
RPS6KB1 P23443 1/20 0.39
AURKB Q96GD4 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9736989 0.87 CYP2D6 (0.40) CYP2D6CASRMETAP2METAP1AURKA
SCHEMBL9738323 0.84 KDM4E (0.56) SCN1ASCN5ASCN8ACYP2D6CASR
SCHEMBL9738556 0.82 SCN1A (0.41) SCN1ASCN5ASCN8AMEN1KMT2A
SCHEMBL9739881 0.82 SCN1A (0.40) SCN1ASCN5ASCN8ACYP2D6CASR
SCHEMBL9737123 0.75 CA2 (0.45) MEN1KMT2ACA1CA2
SCHEMBL573694 0.71 PKM (0.44) CYP2D6CA1CA2
SCHEMBL30944279 0.71 PTGER4 (0.55) MEN1KMT2AAURKARPS6KB1AURKB
SCHEMBL28519320 0.71 PTGER4 (0.55) MEN1KMT2AAURKARPS6KB1AURKB
SCHEMBL28519323 0.71 PTGER4 (0.55) MEN1KMT2AAURKARPS6KB1AURKB
SCHEMBL9737103 0.70 CA2 (0.39) MEN1KMT2ACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5145867-A NAPHTHYLALKYLAMINO-SUBSTITUTED SULFAMOYLBENZOIC ACID DERIVATIVES, AND THE USE THEREOF AS MEDICINES HOECHST AKTIENGESELLSCHAFT (DE) 1992-09-08 US disclosed