SCHEMBL9738909

SCHEMBL9738909

COc1cc2c(cc1OC)CC(=O)N(CC1CCCCN(Cc3ccccc3)C1)C=C2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 3/20 0.44
ACHE P22303 2/20 0.43
BACE1 P56817 2/20 0.43
FAAH O00519 1/20 0.43
ABCC4 O15439 1/20 0.43
CACNA1F O60840 1/20 0.43
PDE5A O76074 1/20 0.43
ABCB11 O95342 1/20 0.43
APP P05067 1/20 0.43
CHRM2 P08172 1/20 0.43
ABCB1 P08183 1/20 0.43
CYP3A4 P08684 1/20 0.43
CHRM5 P08912 1/20 0.43
ADRA2A P08913 1/20 0.43
CHRM1 P11229 1/20 0.43
ADRA2C P18825 1/20 0.43
DRD4 P21917 1/20 0.43
SLC6A2 P23975 1/20 0.43
MAOB P27338 1/20 0.43
AGTR1 P30556 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9738933 0.97 BCHE (0.45) BCHEACHEBACE1FAAHABCC4
SCHEMBL9214964 0.82 CHRNB4 (0.41) PDE4DBRD4
SCHEMBL9740380 0.81 HCN4 (0.54) SIGMAR1BRD4
SCHEMBL9739668 0.81 HCN4 (0.54) SIGMAR1BRD4
Hydrochloric Acid SCHEMBL10766227 0.81 HCN4 (0.53) CYP3A4BRD4
SCHEMBL9212352 0.80 ACHE (0.43) BCHEACHEDRD4BRD4
SCHEMBL9739274 0.80 CHRNB4 (0.44) PDE4DBRD4
SCHEMBL9739670 0.78 HCN4 (0.55) ABCB1CYP3A4BRD4
SCHEMBL9215863 0.76 BRD4 (0.40) ACHECHRM2ABCB1CHRM1PDE4D
Hydrochloric Acid SCHEMBL9739548 0.75 MAOA (0.36) ACHECYP3A4MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0224794-B1 CYCLIC AMINE DERIVATIVES, MEDICINES CONTAINING THESE COMPOUNDS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1990-09-12 EP disclosed
EP-0224794-A2 Cyclic amine derivatives, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-06-10 EP disclosed