SCHEMBL9739825

SCHEMBL9739825

N#CC1(C#N)OC1c1cccc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
THRB P10828 2/20 0.36
HTT P42858 2/20 0.36
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
HPGD P15428 1/20 0.36
IDO1 P14902 1/20 0.36
TDO2 P48775 1/20 0.36
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
HTR2B P41595 2/20 0.36
KDM1A O60341 1/20 0.36
RCOR1 Q9UKL0 1/20 0.36
TSHR P16473 1/20 0.35
MCL1 Q07820 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10703931 0.80 MAPT (0.42) TAAR1MEN1KMT2AALDH1A1MAPT
SCHEMBL9738560 0.77 ALDH1A1 (0.38) MEN1KMT2AALDH1A1MAPTTHRB
SCHEMBL17684664 0.69 TAAR1 (0.40) TAAR1HTR2AHTR2CHTR2BKDM1A
SCHEMBL9059555 0.68 CHRNB2 (0.36) MEN1KMT2AALDH1A1HPGD
SCHEMBL31075268 0.67 KDM1A (0.47) TAAR1MEN1KMT2AALDH1A1MAPT
Cyanamide SCHEMBL27345527 0.66 ALDH1A1 (0.52) TAAR1MEN1KMT2AALDH1A1MAPT
SCHEMBL17735939 0.66 KDM1A (0.39) TAAR1ALDH1A1MAPTTHRBHTT
SCHEMBL17728209 0.66 TAAR1 (0.37) TAAR1HTR2AHTR2CHTR2BKDM1A
SCHEMBL15327483 0.65 TAAR1 (0.44) TAAR1MEN1KMT2AALDH1A1MAPT
SCHEMBL17684167 0.65 HSD11B1 (0.39) TAAR1HTR2AHTR2CHTR2BKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5082842-A Sedatives HOFFMANN-LA ROCHE INC. (US) 1992-01-21 US disclosed
US-4889854-A MUSCLE RELAXANT, SEDATIVE-HYPNOTIC, ANXIOLYTIC AND-OR ANTICONVULSANT ACTIVITY HOFFMAN-LA ROCHE INC. (US) 1989-12-26 US disclosed
EP-0294599-A2 Tricyclic pyridone derivatives F. HOFFMANN-LA ROCHE AG (CH) 1988-12-14 EP disclosed