SCHEMBL9740598

SCHEMBL9740598

Nc1c(Cl)cc(COc2ccc3[nH][c]cc3c2)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.39
MAOB P27338 5/20 0.38
ALOX5 P09917 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
SRD5A2 P31213 1/20 0.36
HSD17B10 Q99714 1/20 0.36
NOS1 P29475 3/20 0.36
NOS3 P29474 2/20 0.36
NOS2 P35228 1/20 0.36
MAOA P21397 1/20 0.34
HTR1A P08908 1/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
TEC P42680 1/20 0.34
PDGFRB P09619 1/20 0.34
PDGFRA P16234 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL694423 0.78 ALOX5 (0.62) MAOBALOX5KDM4EALDH1A1CYP1A2
SCHEMBL9741209 0.76 MAOB (0.36) CYP2D6MAOBKDM4ENOS1NOS3
SCHEMBL9740058 0.75 MAPT (0.37) KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9740778 0.74 ALOX5 (0.36) MAOBALOX5MAOAF2
SCHEMBL1388250 0.67 MAOA (0.50) MAOBMAOA
SCHEMBL9740911 0.65 TUBB1 (0.57) MAOBKDM4EALDH1A1HPGD
SCHEMBL315575 0.65 AXL (0.53) KDM4EALDH1A1CYP1A2HPGDHSD17B10
SCHEMBL6840901 0.63 MRGPRX4 (0.50) CYP2D6MAOBMAOA
SCHEMBL5830621 0.62 KDM4E (0.58) KDM4EALDH1A1MAOAPDGFRBPDGFRA
SCHEMBL2971940 0.62 MEN1 (0.47) KDM4EALDH1A1HPGDHSD17B10MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed