SCHEMBL9744937

SCHEMBL9744937

CCOC(=O)C(/C=C/CP(=O)(OCC)OCC)NC=O

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.32
PPARD Q03181 1/20 0.32
TSHR P16473 2/20 0.32
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP3A4 P08684 1/20 0.30
ALOX15 P16050 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10717181 0.77 TSHR (0.36) PPARDTSHR
SCHEMBL9744853 0.77 GAA (0.33) MAPTTSHRCYP2D6CYP2C9CYP2C19
SCHEMBL9744920 0.76 CYP2D6 (0.43) PPARDTSHRCYP2D6CYP2C9CYP2C19
SCHEMBL9745133 0.73 CYP2D6 (0.32) PPARDTSHRCYP2D6CYP2C9CYP2C19
SCHEMBL10913361 0.72 MGAM (0.39) TSHRCYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL9792736 0.72 MGAM (0.39) TSHRCYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL10998341 0.71 MGAM (0.38) TSHRCYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL12226250 0.70 L3MBTL1 (0.38) PPARDTSHRALDH1A1CYP3A4ALOX15
SCHEMBL9840702 0.69
SCHEMBL687973 0.68 MAPT (0.47) MAPTHTTPPARDTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175344-A Anticonvulsants, anxiolytic agents CIBA-GEIGY CORPORATION (US) 1992-12-29 US disclosed
EP-0233154-B1 UNSATURATED AMINO-ACIDS CIBA-GEIGY AG (CH) 1991-12-18 EP disclosed
US-5051413-A For treatment of ischemia, antispasmodic agents, anticonvulsants and anxiety or manic conditions CIBA-GEIGY CORPORATION (US) 1991-09-24 US disclosed
EP-0233154-A2 Unsaturated amino-acids CIBA-GEIGY AG (CH) 1987-08-19 EP disclosed