SCHEMBL9745156

SCHEMBL9745156

CCOC(=O)C1=CN(C=Cc2ccc(O)c(OC)c2)C(C)=C(C(=O)OC)C1c1cccc(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 7/20 0.43
MAOB P27338 2/20 0.43
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 3/20 0.41
HSD17B10 Q99714 3/20 0.41
CASP1 P29466 2/20 0.41
CASP7 P55210 2/20 0.41
MAPT P10636 4/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
ACHE P22303 1/20 0.41
MAPK1 P28482 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
GLA P06280 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PDE4B Q07343 1/20 0.39
PDE4D Q08499 1/20 0.39
CXCL12 P48061 1/20 0.39
AR P10275 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9745284 0.86 KMT2A (0.37) GAAKDM4EALDH1A1HSD17B10CASP1
SCHEMBL9745152 0.77 CACNA1B (0.51) KDM4EALDH1A1HSD17B10MAPTKMT2A
SCHEMBL9745992 0.71 PDE4B (0.47) GAAMAPTKMT2AMEN1MAPK1
SCHEMBL14262742 0.70 ADORA3 (0.51) GAAKDM4EALDH1A1HSD17B10MAPT
SCHEMBL10515946 0.68 CYP1A2 (0.62) MAPTKMT2AMEN1MAPK1NPSR1
SCHEMBL9745148 0.67 ADORA3 (0.48) GAAKDM4EALDH1A1HSD17B10MAPT
SCHEMBL9502243 0.66 ADORA3 (0.73) GAAKDM4EALDH1A1HSD17B10MAPT
SCHEMBL11877354 0.65 CACNA1F (0.54) MAPTKMT2AMEN1ACHEMAPK1
SCHEMBL30568635 0.64 KDM1A (0.76) MAOBALDH1A1MAPTKMT2AMEN1
SCHEMBL11771981 0.64 KDM4E (0.52) GAAKDM4EALDH1A1HSD17B10CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0215250-B1 2-SUBSTITUTED-1,4-DIHYDROPYRIDINES, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1992-12-30 EP disclosed
US-4845113-A USEFUL IN RADICAL SCAVENGING THERAPY BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1989-07-04 US disclosed
EP-0215250-A1 2-Substituted-1,4-dihydropyridines, method for their preparation and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1987-03-25 EP disclosed