SCHEMBL9745148

SCHEMBL9745148

C=C(C1=C(C(=O)OCC)C(c2cccc(Cl)c2)C(C(=O)OC)=C(C)N1)c1ccc(O)c(OC)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.48
HIF1A Q16665 5/20 0.48
CYP2C9 P11712 5/20 0.48
MEN1 O00255 4/20 0.48
CYP1A2 P05177 4/20 0.48
CYP3A4 P08684 4/20 0.48
CYP2C19 P33261 4/20 0.48
KMT2A Q03164 4/20 0.48
MAPT P10636 3/20 0.48
LMNA P02545 2/20 0.48
CYP2D6 P10635 2/20 0.48
TSHR P16473 2/20 0.48
NFKB1 P19838 2/20 0.48
THPO P40225 2/20 0.48
POLB P06746 1/20 0.48
MAPK1 P28482 1/20 0.48
GPR55 Q9Y2T6 1/20 0.48
CACNA1B Q00975 7/20 0.45
HSD17B2 P37059 1/20 0.45
KDM4E B2RXH2 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9745272 0.84 HIF1A (0.45) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL9502243 0.81 ADORA3 (0.73) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL9745152 0.80 CACNA1B (0.51) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL11771568 0.79 ABCC1 (0.61) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL3026966 0.76 ABCC1 (0.71) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL9744733 0.76 CACNA1B (0.55) ADORA3CACNA1BCACNA1FCACNA1DCACNA1S
SCHEMBL3028393 0.74 GAA (0.66) ADORA3MEN1KMT2AMAPTLMNA
SCHEMBL11773488 0.73 CACNA1F (0.56) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL9501260 0.73 ADORA3 (0.57) ADORA3HIF1ACYP2C9MEN1CYP1A2
SCHEMBL7349302 0.73 ADORA3 (0.64) ADORA3HIF1ACYP2C9MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0215250-B1 2-SUBSTITUTED-1,4-DIHYDROPYRIDINES, METHOD FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1992-12-30 EP disclosed
US-4845113-A USEFUL IN RADICAL SCAVENGING THERAPY BOEHRINGER BIOCHEMIA ROBIN S.P.A. (IT) 1989-07-04 US disclosed
EP-0215250-A1 2-Substituted-1,4-dihydropyridines, method for their preparation and pharmaceutical compositions containing them BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1987-03-25 EP disclosed