SCHEMBL9747658

SCHEMBL9747658

N#Cc1ccc2c(ccc3[nH]c(=O)c(=O)[nH]c32)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 1/20 0.47
IMPDH1 P20839 1/20 0.47
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
FASN P49327 1/20 0.44
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42
CYP19A1 P11511 1/20 0.41
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
AR P10275 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
CHEK1 O14757 1/20 0.38
CCNE2 O96020 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30905530 0.76 NOS3 (0.53) IMPDH2IMPDH1FASNGRIN2DGRIN3B
SCHEMBL118018 0.76 NOS3 (0.53) IMPDH2IMPDH1FASNGRIN2DGRIN3B
SCHEMBL28489960 0.73 GRM5 (0.64) IMPDH2IMPDH1CA1CA2CHEK1
SCHEMBL13037656 0.73 CA2 (0.55) IMPDH2IMPDH1CA1CA2CYP19A1
SCHEMBL1054605 0.73 CA12 (0.56) IMPDH2IMPDH1CA1CA2FASN
SCHEMBL29891877 0.72 IMPDH2 (0.51) IMPDH2IMPDH1CA1CA2FASN
Hydrochloric Acid SCHEMBL7004520 0.72 GRM5 (0.62) IMPDH2IMPDH1CA1CA2CHEK1
SCHEMBL9747072 0.72 GRIN2D (0.63) FASNGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL12310183 0.71 CA2 (0.53) IMPDH2IMPDH1CA1CA2CYP19A1
SCHEMBL12320904 0.71 CA2 (0.53) IMPDH2IMPDH1CA1CA2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0511152-A2 Quinoxaline compounds, their preparation and use NOVO NORDISK A/S (DK) 1992-10-28 EP disclosed