SCHEMBL9749343

SCHEMBL9749343

CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CCN(C)CC3CO)c(F)c21

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 0.61
ALDH1A1 P00352 8/20 0.61
HPGD P15428 7/20 0.61
HSD17B10 Q99714 7/20 0.61
PMP22 Q01453 1/20 0.60
DRD3 P35462 1/20 0.52
MEN1 O00255 1/20 0.48
NPC1 O15118 1/20 0.48
KMT2A Q03164 1/20 0.48
LMNA P02545 2/20 0.46
BRD4 O60885 1/20 0.46
TSHR P16473 1/20 0.46
HTT P42858 1/20 0.46
CYP2J2 P51589 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
ALB P02768 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
ADRA2B P18089 1/20 0.45
MAPK1 P28482 1/20 0.45
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10425073 0.92 KDM4E (0.70) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9749882 0.86 KDM4E (0.51) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9749353 0.86 KCNH2 (0.55) KDM4EALDH1A1HPGDHSD17B10ALB
SCHEMBL9749919 0.85 KDM4E (0.61) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9749304 0.83 LMNA (0.53) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL312380 0.83 KDM4E (0.84) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL10425075 0.81 KDM4E (0.64) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL10425078 0.81 KDM4E (0.64) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL10621416 0.80 KDM4E (0.68) KDM4EALDH1A1HPGDHSD17B10PMP22
SCHEMBL9837564 0.80 KDM4E (0.62) KDM4EALDH1A1HPGDHSD17B10PMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0216345-B1 QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1992-02-19 EP disclosed
US-4977265-A WITH BACTERICIDAL ACTIVITY HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed
US-4946847-A BACTERICIDES HOFFMANN-LA ROCHE INC. (US) 1990-08-07 US disclosed
US-4806541-A ANTIBACTERIAL AGENTS HOFFMANN-LA ROCHE INC. (US) 1989-02-21 US disclosed
EP-0216345-A2 Quinoline derivatives F. HOFFMANN-LA ROCHE AG (CH) 1987-04-01 EP disclosed