SCHEMBL9749563

SCHEMBL9749563

COc1ccc(-n2nc(C(=O)CCC(=O)N(C)O)cc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.73
ALOX5 P09917 2/20 0.73
MALT1 Q9UDY8 6/20 0.64
MARS1 P56192 1/20 0.57
CHRNA7 P36544 2/20 0.55
RPA1 P27694 3/20 0.54
CCKAR P32238 2/20 0.53
PTGS1 P23219 4/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
NFKB1 P19838 2/20 0.53
NFKB2 Q00653 2/20 0.53
RELA Q04206 2/20 0.53
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
TSHR P16473 1/20 0.52
CYP2C19 P33261 1/20 0.52
THPO P40225 1/20 0.52
BLM P54132 1/20 0.52
PMP22 Q01453 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9149353 0.91 PTGS2 (0.60) PTGS2ALOX5MALT1CHRNA7RPA1
SCHEMBL8475502 0.89 MALT1 (0.68) PTGS2ALOX5MALT1MARS1CHRNA7
Tepoxalin SCHEMBL75441 0.84 PTGS2 (1.00) PTGS2ALOX5MALT1CCKARPTGS1
Tepoxalin SCHEMBL9519652 0.84 PTGS2 (0.98) PTGS2ALOX5MALT1CCKARPTGS1
SCHEMBL9080028 0.82 PTGS2 (0.81) PTGS2ALOX5MALT1CCKARPTGS1
SCHEMBL9353410 0.81 CHRNA7 (0.72) PTGS2ALOX5MALT1MARS1CHRNA7
Tepoxalin SCHEMBL28256087 0.79 ALOX5 (0.87) PTGS2ALOX5MALT1CCKARPTGS1
SCHEMBL9349921 0.79 PTGS2 (0.66) PTGS2ALOX5MALT1MARS1CCKAR
SCHEMBL9522439 0.78 PTGS2 (0.79) PTGS2ALOX5MALT1CCKARPTGS1
Water SCHEMBL9349800 0.78 PTGS2 (0.65) PTGS2ALOX5MALT1CCKARPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5117054-A Chemical intermediate for antiinflammatory agents ORTHO PHARMACEUTICAL CORPORATION (US) 1992-05-26 US disclosed