SCHEMBL8475502

SCHEMBL8475502

COc1ccc(-n2nc(C(=O)CCC(=O)O)cc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 4/20 0.68
MARS1 P56192 1/20 0.63
RPA1 P27694 3/20 0.60
RXRA P19793 1/20 0.60
RXRB P28702 1/20 0.60
RXRG P48443 1/20 0.60
PTGS2 P35354 3/20 0.59
ALOX5 P09917 1/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
CCKAR P32238 5/20 0.58
CHRNA7 P36544 2/20 0.58
PPP1CA P62136 1/20 0.57
PTGS1 P23219 2/20 0.55
NFKB1 P19838 1/20 0.55
NFKB2 Q00653 1/20 0.55
RELA Q04206 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9749563 0.89 PTGS2 (0.73) MALT1MARS1RPA1PTGS2ALOX5
SCHEMBL5393447 0.83 RXRA (0.84) MALT1RXRARXRBRXRGPTGS2
SCHEMBL9353410 0.81 CHRNA7 (0.72) MALT1MARS1RPA1PTGS2ALOX5
SCHEMBL9056282 0.80 RPA1 (0.90) MALT1MARS1RPA1SMN1; SMN2CHRNA7
SCHEMBL9149353 0.79 PTGS2 (0.60) MALT1RPA1PTGS2ALOX5CCKAR
SCHEMBL3262361 0.78 CHRNA7 (0.72) MALT1MARS1RPA1PTGS2CCKAR
SCHEMBL117493 0.77 MARS1 (1.00) MALT1MARS1RPA1SMN1; SMN2PPP1CA
SCHEMBL9349843 0.77 CCKAR (0.60) MALT1MARS1RXRARXRBRXRG
SCHEMBL9519465 0.77 PTGS2 (0.79) MALT1MARS1RXRARXRBRXRG
SCHEMBL9349407 0.76 SMN1; SMN2 (0.63) MALT1MARS1RPA1PTGS2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5869674-A DI-2-((1,5,4-SUBSTITUTED)-PYRAZOL-3-YL) ETHYLCARBONATE, WITH AT LEAST ONE 2-QUINOLINYLMETHOXYPHENYL GROUP ON PYRAZOL ORTHO PHARMACEUTICAL CORPORATION (US) 1999-02-09 US disclosed
US-5843958-A Arylpyrazoles as leukotriene inhibitors ORTHO PHARMACEUTICAL CORPORATION (US) 1998-12-01 US disclosed