SCHEMBL9149353

SCHEMBL9149353

COc1ccc(-n2nc(C(=O)CCC(=O)N(C)O)cc2-c2ccc(C)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.60
ALOX5 P09917 1/20 0.60
CHRNA7 P36544 1/20 0.56
RPA1 P27694 1/20 0.55
PTGS1 P23219 1/20 0.54
CCKAR P32238 3/20 0.52
MALT1 Q9UDY8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9749563 0.91 PTGS2 (0.73) PTGS2ALOX5CHRNA7RPA1PTGS1
SCHEMBL9520508 0.84 ALOX5 (0.83) PTGS2ALOX5PTGS1CCKAR
SCHEMBL9350647 0.81 CA9 (0.71) CHRNA7RPA1CCKARMALT1
SCHEMBL9349395 0.80 RPA1 (0.64) CHRNA7RPA1CCKARMALT1
SCHEMBL8475502 0.79 MALT1 (0.68) PTGS2ALOX5CHRNA7RPA1PTGS1
SCHEMBL9054421 0.78 CA9 (0.65) PTGS2CHRNA7RPA1MALT1
SCHEMBL9349936 0.77 RPA1 (0.70) CHRNA7RPA1CCKARMALT1
SCHEMBL9349904 0.77 RPA1 (0.49) PTGS2ALOX5RPA1CCKARMALT1
SCHEMBL9349431 0.77 RPA1 (0.49) PTGS2ALOX5RPA1CCKARMALT1
SCHEMBL9056282 0.76 RPA1 (0.90) CHRNA7RPA1MALT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380869-A Regioselective synthesis of 1,5-diaryl pyrazole anti-inflammatory agents ORTHO PHARMACEUTICAL CORPORATION (US) 1995-01-10 US disclosed
US-5260458-A 2-oxo tetrahydrofuran compounds ORTHO PHARMACEUTICAL CORPORATION (US) 1993-11-09 US disclosed
EP-0534800-A2 Regioselective synthesis of 1,5-diaryl pyrazole anti-inflammatory agents ORTHO PHARMACEUTICAL CORPORATION (US) 1993-03-31 EP disclosed
US-5117054-A Chemical intermediate for antiinflammatory agents ORTHO PHARMACEUTICAL CORPORATION (US) 1992-05-26 US disclosed