SCHEMBL9750232

SCHEMBL9750232

O=C=NC(=O)c1ccc2cnccc2c1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.45
CYP3A4 P08684 6/20 0.43
HIPK2 Q9H2X6 1/20 0.42
KDM2B Q8NHM5 1/20 0.41
IMPDH2 P12268 3/20 0.41
AKT1 P31749 4/20 0.41
AR P10275 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
FASN P49327 1/20 0.38
CDK2 P24941 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28486284 0.82 HIPK2 (0.53) SMYD3CYP3A4HIPK2KDM2BIMPDH2
SCHEMBL9160200 0.78 CES2 (0.57) CYP3A4
SCHEMBL19900296 0.77 SMYD3 (0.44) SMYD3CYP3A4HIPK2KDM2BIMPDH2
SCHEMBL113378 0.76 SMYD3 (0.55) SMYD3CYP3A4HIPK2KDM2BIMPDH2
SCHEMBL29489099 0.76 SMYD3 (0.55) SMYD3CYP3A4HIPK2KDM2BIMPDH2
Hydrochloric Acid SCHEMBL7557776 0.75 SMYD3 (0.54) SMYD3CYP3A4HIPK2KDM2BIMPDH2
SCHEMBL12765931 0.75 SMYD3 (0.50) SMYD3CYP3A4HIPK2KDM2BIMPDH2
SCHEMBL3126130 0.75 IMPDH2 (0.53) SMYD3CYP3A4HIPK2KDM2BIMPDH2
SCHEMBL29522657 0.75 AR (0.62) SMYD3CYP3A4HIPK2KDM2BIMPDH2
SCHEMBL4280154 0.75 AR (0.62) SMYD3CYP3A4HIPK2KDM2BIMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0234098-B1 N-[piperidylaminocarbonyl]quinolinecarboxamide derivatives having psychotropic activity JOHN WYETH & BROTHER LIMITED (GB) 1992-02-26 EP disclosed
US-4778802-A PSYCHOTROPIC ACTIVITY; ANTIDEPRESSANTS JOHN WYETH & BROTHER, LTD. (GB) 1988-10-18 US disclosed
EP-0234098-A1 N-[piperidylaminocarbonyl]quinolinecarboxamide derivatives having psychotropic activity JOHN WYETH & BROTHER LIMITED (GB) 1987-09-02 EP disclosed