SCHEMBL9752001

SCHEMBL9752001

N[C@@H](CC(=O)O)C(=O)N[C@H](CO)Cc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.62
CYP3A4 P08684 1/20 0.62
CTSC P53634 2/20 0.52
SLC15A1 P46059 1/20 0.49
MC4R P32245 1/20 0.48
MC3R P41968 1/20 0.48
ALPI P09923 1/20 0.47
PKM P14618 1/20 0.47
PTGS1 P23219 1/20 0.47
XIAP P98170 1/20 0.47
SLC7A5 Q01650 1/20 0.47
LTA4H P09960 5/20 0.47
ROCK2 O75116 1/20 0.47
RPS6KA5 O75582 1/20 0.47
RPS6KA4 O75676 1/20 0.47
PRKACA P17612 1/20 0.47
GSK3A P49840 1/20 0.47
GSK3B P49841 1/20 0.47
IRAK1 P51617 1/20 0.47
PRKX P51817 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27182846 1.00 MAPK1 (0.62) MAPK1CYP3A4CTSCSLC15A1MC4R
SCHEMBL7457031 1.00 MAPK1 (0.62) MAPK1CYP3A4CTSCSLC15A1MC4R
SCHEMBL24453079 0.91 MAPK1 (0.69) MAPK1CYP3A4CTSCSLC15A1MC4R
SCHEMBL13669592 0.91 MAPK1 (0.69) MAPK1CYP3A4CTSCSLC15A1MC4R
SCHEMBL27182753 0.89 SLC7A5 (0.50) MAPK1CYP3A4SLC7A5
SCHEMBL27471057 0.86 CYP3A4 (0.68) MAPK1CYP3A4CTSCLTA4H
SCHEMBL12228016 0.83 CYP3A4 (0.47) MAPK1CYP3A4CTSCSLC15A1SLC7A5
SCHEMBL10558069 0.82 MAPK1 (0.75) MAPK1CYP3A4CTSCROCK2RPS6KA5
SCHEMBL11039145 0.82 OPRD1 (0.53) CTSCMC4RMC3RSLC7A5
SCHEMBL10632506 0.81 SLC15A1 (0.58) CTSCSLC15A1ALPIPKMPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0449884-A4 DERIVATIVES OF TETRAPEPTIDES AS CCK AGONISTS 1991-10-30 EP disclosed
EP-0449884-A1 DERIVATIVES OF TETRAPEPTIDES AS CCK AGONISTS ABBOTT LABORATORIES (US) 1991-10-09 EP disclosed