SCHEMBL9753008

SCHEMBL9753008

CC(C)c1c(C=CC=O)c(-c2ccc(F)cc2)nn2c(Cl)cc(Cl)c12

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.32
KDM5B Q9UGL1 1/20 0.32
MAPK14 Q16539 1/20 0.31
KMT2A Q03164 1/20 0.30
PTGS1 P23219 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753006 1.00 PTGS2 (0.32) PTGS2KDM5BMAPK14KMT2APTGS1
SCHEMBL9753228 0.83 MAPK14 (0.39) PTGS2KDM5BMAPK14KMT2APTGS1
SCHEMBL9753226 0.83 MAPK14 (0.39) PTGS2KDM5BMAPK14KMT2APTGS1
SCHEMBL9753676 0.82 PTGS2 (0.37) PTGS2KDM5BMAPK14KMT2A
SCHEMBL9753671 0.82 PTGS2 (0.37) PTGS2KDM5BMAPK14KMT2A
SCHEMBL9753232 0.82 MAPK14 (0.33) PTGS2KDM5BMAPK14KMT2A
SCHEMBL9753231 0.82 MAPK14 (0.33) PTGS2KDM5BMAPK14KMT2A
SCHEMBL9753292 0.79 HMGCR (0.41)
SCHEMBL9753286 0.79 HMGCR (0.41)
SCHEMBL9753035 0.78 AKT1 (0.36) PTGS2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed