SCHEMBL9753063

SCHEMBL9753063

CC(C)c1c(C=O)c(-c2ccccc2)nn2cccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.39
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
ADORA2A P29274 3/20 0.37
KMT2A Q03164 2/20 0.37
ADORA1 P30542 2/20 0.37
MIF P14174 2/20 0.37
MEN1 O00255 1/20 0.37
PDE5A O76074 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
PDE4A P27815 1/20 0.37
CYP2C19 P33261 1/20 0.37
BLM P54132 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753321 0.88 MAPK14 (0.44) EGFRALDH1A1ADORA2AKMT2AADORA1
SCHEMBL9753122 0.87 EGFR (0.38) EGFRALDH1A1ADORA2AKMT2AADORA1
SCHEMBL9753124 0.87 EGFR (0.38) EGFRALDH1A1ADORA2AKMT2AADORA1
SCHEMBL9753354 0.83 PTGS2 (0.34) EGFRALDH1A1ADORA2AKMT2AADORA1
SCHEMBL15070164 0.81 EGFR (0.44) EGFRALDH1A1ADORA2AKMT2AADORA1
SCHEMBL8811759 0.81 ADORA2A (0.45) EGFRALDH1A1LMNAADORA2AADORA1
SCHEMBL9753040 0.80 PTGS2 (0.36) EGFRALDH1A1ADORA2AADORA1KCNH2
SCHEMBL9753160 0.77 MAPK14 (0.41) EGFRALDH1A1ADORA2AKMT2AADORA1
SCHEMBL9753157 0.77 MAPK14 (0.41) EGFRALDH1A1ADORA2AKMT2AADORA1
SCHEMBL9752941 0.77 ALDH1A1 (0.35) EGFRALDH1A1ADORA2AADORA1PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed