SCHEMBL9753040

SCHEMBL9753040

CC(C)c1c(C=O)c(-c2ccc(F)c(Cl)c2)nn2cccc12

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.36
EGFR P00533 2/20 0.36
PGR P06401 1/20 0.35
KDR P35968 1/20 0.35
MAPK14 Q16539 1/20 0.35
PTGS1 P23219 3/20 0.33
TGFBR1 P36897 4/20 0.33
TGFBR2 P37173 2/20 0.33
HTR6 P50406 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
SPR P35270 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753354 0.90 PTGS2 (0.34) PTGS2EGFRPGRKDRMAPK14
SCHEMBL9752932 0.90 PTGS2 (0.34) PTGS2EGFRPGRKDRMAPK14
SCHEMBL9752930 0.90 PTGS2 (0.34) PTGS2EGFRPGRKDRMAPK14
SCHEMBL9753321 0.84 MAPK14 (0.44) PTGS2EGFRMAPK14PTGS1ADORA2A
SCHEMBL27438905 0.82 RORC (0.38) EGFRPGRKDRTGFBR1TGFBR2
SCHEMBL9753400 0.80 TP53 (0.36) EGFRMAPK14ADORA2AADORA1SPR
SCHEMBL9753002 0.80 TGFBR1 (0.36) PTGS2EGFRPGRKDRMAPK14
SCHEMBL9753063 0.80 EGFR (0.39) PTGS2EGFRMAPK14ADORA2AADORA1
SCHEMBL9753724 0.80 PTGS2 (0.32) PTGS2EGFRPGRMAPK14ADORA2A
SCHEMBL9753721 0.80 PTGS2 (0.32) PTGS2EGFRPGRMAPK14ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed
CN-1056690-A PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO (JP) 1991-12-04 CN disclosed