SCHEMBL9753354

SCHEMBL9753354

CC(C)c1c(C=O)c(-c2ccc(F)c(F)c2)nn2cccc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.34
EGFR P00533 3/20 0.33
PIK3CD O00329 2/20 0.33
ABL1 P00519 2/20 0.33
HCK P08631 2/20 0.33
SRC P12931 2/20 0.33
KDR P35968 2/20 0.33
PIK3CA P42336 2/20 0.33
PIK3CB P42338 2/20 0.33
MTOR P42345 2/20 0.33
PIK3CG P48736 2/20 0.33
EPHB4 P54760 2/20 0.33
PRKDC P78527 2/20 0.33
MAPK14 Q16539 2/20 0.32
ADORA2A P29274 2/20 0.32
ADORA1 P30542 2/20 0.32
PGR P06401 1/20 0.32
RAF1 P04049 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2B P29275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753040 0.90 PTGS2 (0.36) PTGS2EGFRKDRMAPK14ADORA2A
SCHEMBL9753724 0.89 PTGS2 (0.32) PTGS2EGFRMAPK14ADORA2AADORA1
SCHEMBL9753721 0.89 PTGS2 (0.32) PTGS2EGFRMAPK14ADORA2AADORA1
SCHEMBL9753321 0.87 MAPK14 (0.44) PTGS2EGFRMAPK14ADORA2AADORA1
SCHEMBL9753063 0.83 EGFR (0.39) PTGS2EGFRMAPK14ADORA2AADORA1
SCHEMBL9752941 0.81 ALDH1A1 (0.35) PTGS2EGFRMAPK14ADORA2AADORA1
SCHEMBL9752932 0.80 PTGS2 (0.34) PTGS2EGFRKDRMAPK14ADORA2A
SCHEMBL9752930 0.80 PTGS2 (0.34) PTGS2EGFRKDRMAPK14ADORA2A
SCHEMBL9753346 0.79 GCGR (0.39) EGFRMAPK14ADORA2AADORA1RAF1
SCHEMBL9753639 0.77 HMGCR (0.34) PTGS2PGRADORA3ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed