SCHEMBL9753176

SCHEMBL9753176

COc1ccc(CCN2CCCC2CN=S(=O)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 5/20 0.53
TRPV6 Q9H1D0 1/20 0.51
DRD2 P14416 1/20 0.44
FKBP1A P62942 2/20 0.43
ALDH1A1 P00352 1/20 0.43
POLB P06746 1/20 0.43
TSHR P16473 1/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753177 1.00 HRH3 (0.53) HRH3TRPV6DRD2FKBP1AALDH1A1
SCHEMBL9739334 0.84 TRPV6 (0.59) HRH3TRPV6DRD2FKBP1AALDH1A1
SCHEMBL9668361 0.75 HRH3 (0.50) HRH3DRD2FKBP1AALDH1A1POLB
SCHEMBL9668366 0.75 HRH3 (0.50) HRH3DRD2FKBP1AALDH1A1POLB
SCHEMBL9372067 0.75 HRH3 (0.68) HRH3TRPV6
SCHEMBL9374317 0.75 HRH3 (0.68) HRH3TRPV6
SCHEMBL9372055 0.75 HRH3 (0.68) HRH3TRPV6
SCHEMBL9669966 0.74 ALDH1A1 (0.47) HRH3FKBP1AALDH1A1POLBTSHR
SCHEMBL9376275 0.73 HRH3 (0.65) HRH3TRPV6
SCHEMBL9372378 0.73 HRH3 (0.65) HRH3TRPV6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991010648-A1 DIPHENYLSULPHOXIMINE MUSCARINIC RECEPTOR ANTAGONISTS PFIZER LIMITED (GB) 1991-07-25 WO disclosed