SCHEMBL9754150

SCHEMBL9754150

CC(C)Cc1ccc(Cc2nc(O)c(-c3ccccc3)s2)cc1

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 5/20 0.48
XIAP P98170 1/20 0.41
PTGDR2 Q9Y5Y4 2/20 0.41
KDM4E B2RXH2 1/20 0.39
PTGS2 P35354 1/20 0.39
DHODH Q02127 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9754002 0.88 ALOX5 (0.47) ALOX5PTGS2DHODHKMT2A
SCHEMBL9754030 0.86 ALOX5 (0.44) ALOX5PTGS2KMT2A
SCHEMBL9754000 0.79 ALOX5 (0.46) ALOX5PTGS2
SCHEMBL9754025 0.77 ALOX5 (0.43) ALOX5PTGDR2PTGS2
SCHEMBL9803529 0.76 ALOX5 (0.43) ALOX5PTGDR2PTGS2
SCHEMBL6546976 0.72 CALM1 (0.57) ALOX5PTGS2
SCHEMBL22455579 0.71 HPGD (0.43) KDM4EDHODHMAPTHTTKMT2A
SCHEMBL22455603 0.71 HDAC6 (0.43) KDM4EDHODHMAPTHTTKMT2A
Isobutylbenzene SCHEMBL363626 0.70 TAAR1 (0.61) ALOX5PTGS2
SCHEMBL23954137 0.69 ADORA3 (0.45) ALOX5PTGDR2DHODHMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991008744-A1 THIAZOLE LIPOXYGENASE-INHIBITING COMPOUNDS DERIVED FROM NON-STEROIDAL ANTIINFLAMMATORY CARBOXYLIC ACIDS ABBOTT LABORATORIES (US) 1991-06-27 WO claimed
US-5032588-A Non-steroidal antiinflammatory ABBOTT LABORATORIES (US) 1991-07-16 US disclosed
WO-1991008744-A1 THIAZOLE LIPOXYGENASE-INHIBITING COMPOUNDS DERIVED FROM NON-STEROIDAL ANTIINFLAMMATORY CARBOXYLIC ACIDS ABBOTT LABORATORIES (US) 1991-06-27 WO disclosed