SCHEMBL9754183

SCHEMBL9754183

Cc1oncc1C(=O)N(Cc1ccccc1)c1ccc(CC(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 13/20 0.43
PDK2 Q15119 2/20 0.43
PDK4 Q16654 2/20 0.43
PDK3 Q15120 1/20 0.43
RAB9A P51151 1/20 0.42
ATF1 P18846 1/20 0.42
NFKB1 P19838 1/20 0.42
NR1H4 Q96RI1 1/20 0.42
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.41
CNR2 P34972 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9539254 0.90 RAB9A (0.50) PDK1PDK2PDK4PDK3RAB9A
SCHEMBL8808399 0.88 RAB9A (0.51) PDK1PDK2PDK4PDK3RAB9A
SCHEMBL3049960 0.87 PDK1 (0.52) PDK1PDK2PDK4PDK3RAB9A
SCHEMBL9754181 0.85 NR1H4 (0.43) PDK1PDK2PDK4PDK3RAB9A
SCHEMBL27323811 0.79 LMNA (0.41) RAB9AGAATSHR
SCHEMBL5071880 0.72 RAB9A (0.44) RAB9ATSHR
SCHEMBL9392594 0.72 KMT2A (0.52) RAB9A
SCHEMBL5071947 0.71 NPC1 (0.55) RAB9A
SCHEMBL8810187 0.70 TSHR (0.48) RAB9AGAATSHR
SCHEMBL3059654 0.70 GAA (0.50) PDK1PDK2PDK4PDK3ATF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991017748-A1 ISOXAZOLE-4-CARBOXAMIDES AND HYDROXYALKYLIDENE-CYANOACETAMIDES, DRUGS CONTAINING THESE COMPOUNDS AND USE OF SUCH DRUGS HOECHST AKTIENGESELLSCHAFT (DE) 1991-11-28 WO disclosed