SCHEMBL9539254

SCHEMBL9539254

Cc1oncc1C(=O)N(Cc1ccccc1)c1cccc(CC(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.50
PDK1 Q15118 8/20 0.44
ATF1 P18846 1/20 0.42
NFKB1 P19838 1/20 0.42
S1PR1 P21453 1/20 0.42
S1PR3 Q99500 1/20 0.42
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.41
NPC1 O15118 2/20 0.41
JAK2 O60674 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HTT P42858 1/20 0.41
PAX8 Q06710 1/20 0.41
PDK2 Q15119 1/20 0.41
PDK3 Q15120 1/20 0.41
PDK4 Q16654 1/20 0.41
KMT2A Q03164 1/20 0.41
TSPO P30536 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9754183 0.90 PDK1 (0.43) RAB9APDK1ATF1NFKB1GAA
SCHEMBL3049960 0.87 PDK1 (0.52) RAB9APDK1S1PR1S1PR3GAA
SCHEMBL8808399 0.83 RAB9A (0.51) RAB9APDK1ATF1NFKB1GAA
SCHEMBL9754181 0.80 NR1H4 (0.43) RAB9APDK1ATF1NFKB1GAA
SCHEMBL27323811 0.76 LMNA (0.41) RAB9AGAATSHRNPC1ALDH1A1
SCHEMBL5071880 0.72 RAB9A (0.44) RAB9ATSHRNPC1ALDH1A1HTT
SCHEMBL8810187 0.70 TSHR (0.48) RAB9AGAATSHRNPC1ALDH1A1
SCHEMBL3058600 0.69 RAB9A (0.51) RAB9APDK1ATF1NFKB1GAA
SCHEMBL14300708 0.69 CRHBP (0.43) RAB9ANPC1JAK2ALDH1A1HTT
SCHEMBL3061506 0.69 RAB9A (0.55) RAB9APDK1GAATSHRNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0527736-A1 ISOXAZOLE-4-CARBOXAMIDES AND HYDROXYALKYLIDENE-CYANOACETAMIDES, DRUGS CONTAINING THESE COMPOUNDS AND USE OF SUCH DRUGS. HOECHST AG (DE) 1993-02-24 EP disclosed