SCHEMBL9757062

SCHEMBL9757062

CCOC(=O)c1nc2cccc(O)c2o1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.54
MAOB P27338 1/20 0.54
CA12 O43570 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA7 P43166 1/20 0.53
CA9 Q16790 1/20 0.53
CA14 Q9ULX7 1/20 0.53
NPC1 O15118 2/20 0.48
MAPT P10636 2/20 0.48
RAB9A P51151 1/20 0.48
CYP1A2 P05177 2/20 0.47
KMT2A Q03164 3/20 0.44
MEN1 O00255 2/20 0.44
CYP3A4 P08684 1/20 0.44
GAA P10253 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
RECQL P46063 1/20 0.44
CCR6 P51684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9757020 0.87 FAAH (0.53) MAOAMAOBCA12CA1CA2
SCHEMBL14897791 0.84 ALDH1A1 (0.48) MAOAMAOBCA12CA1CA2
SCHEMBL31745175 0.84 CYP1A2 (0.46) MAOAMAOBCA12CA1CA2
SCHEMBL4346782 0.84 CA12 (0.49) MAOAMAOBCA12CA1CA2
SCHEMBL31745296 0.83 DHODH (0.50) MAOAMAOBMAPTCYP1A2KMT2A
SCHEMBL9757082 0.82 ELANE (0.44) MAOAMAOBCYP1A2KMT2AMEN1
SCHEMBL9757203 0.81 ALDH1A1 (0.41) MAOAMAOBCA12CA1CA2
SCHEMBL9757218 0.80 ALDH1A1 (0.43) NPC1MAPTRAB9ACYP1A2GAA
SCHEMBL29728162 0.79 KDM4E (0.50) NPC1MAPTRAB9ACYP1A2KMT2A
SCHEMBL9760991 0.79 TSHR (0.39) MAOAMAOBCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019475-A2 QUINOLINYL-BENZOHETEROBICYCLIC DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1991-12-26 WO disclosed
US-5041453-A Quinolinyl-benzoheterobicyclic derivatives as antagonists of leukotriene D4 RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-08-20 US disclosed