SCHEMBL9757020

SCHEMBL9757020

CCOC(=O)c1nc2cccc(C)c2o1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.53
CYP1A2 P05177 1/20 0.49
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
LMNA P02545 1/20 0.42
ELANE P08246 1/20 0.42
CETP P11597 1/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9757062 0.87 MAOA (0.54) FAAHCYP1A2MAOAMAOBKMT2A
SCHEMBL31745175 0.86 CYP1A2 (0.46) FAAHCYP1A2MAOAMAOBKMT2A
SCHEMBL14897791 0.86 ALDH1A1 (0.48) FAAHCYP1A2MAOAMAOBKMT2A
SCHEMBL31745296 0.85 DHODH (0.50) CYP1A2MAOAMAOBKMT2AMEN1
SCHEMBL9757082 0.83 ELANE (0.44) FAAHCYP1A2MAOAMAOBKMT2A
SCHEMBL9757218 0.81 ALDH1A1 (0.43) CYP1A2SMN1; SMN2LMNAKDM4EALDH1A1
SCHEMBL29728162 0.80 KDM4E (0.50) CYP1A2KMT2AMEN1SMN1; SMN2LMNA
SCHEMBL38654913 0.79 TRPM8 (0.44) CYP1A2KMT2AMEN1SMN1; SMN2LMNA
SCHEMBL3621004 0.79 RAB9A (0.53) FAAHCYP1A2KMT2ASMN1; SMN2LMNA
SCHEMBL17864533 0.79 CYP1A2 (0.44) CYP1A2MAOAMAOBKMT2ACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019475-A2 QUINOLINYL-BENZOHETEROBICYCLIC DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1991-12-26 WO disclosed
US-5041453-A Quinolinyl-benzoheterobicyclic derivatives as antagonists of leukotriene D4 RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-08-20 US disclosed