SCHEMBL9760013

SCHEMBL9760013

Cn1c(=O)[nH]c2ccc(Cc3ccccc3-n3ccnc3)cc2c1=O

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA2B P29275 1/20 0.42
ADORA1 P30542 1/20 0.42
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6866451 0.80 FNTA (0.48)
SCHEMBL10582405 0.79 GAA (0.40)
SCHEMBL9760033 0.78 SIRT6 (0.39) CA12CA9
SCHEMBL8916747 0.77 TBXAS1 (0.45) CA12CA9
SCHEMBL9190610 0.76 HTR5A (0.38)
SCHEMBL7453705 0.74 HTR5A (0.40)
SCHEMBL669278 0.74 KDM4E (0.46)
SCHEMBL9285801 0.73 IP6K1 (0.51) CA12CA9
SCHEMBL9663508 0.72 IDO1 (0.37)
SCHEMBL9663761 0.72 CYP11B1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5037829-A Antitumor Activity; Androgen, Estrogen Inhibitors; Suppress The Plasma Elimination Of Retinoids JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-06 US claimed
US-5037829-A Antitumor Activity; Androgen, Estrogen Inhibitors; Suppress The Plasma Elimination Of Retinoids JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-06 US disclosed