SCHEMBL9764329

SCHEMBL9764329

Nc1c(Cl)cc(C(O)CN(CCCCCOCCc2ccc(F)cc2)Cc2ccccc2)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.39
SLC2A1 P11166 1/20 0.34
NR1H3 Q13133 4/20 0.34
ADRB1 P08588 1/20 0.34
BCHE P06276 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CYP51A1 Q16850 2/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9764429 0.94 ADRB2 (0.41) ADRB2SLC2A1NR1H3ADRB1BCHE
SCHEMBL9764456 0.94 ADRB2 (0.41) ADRB2SLC2A1NR1H3ADRB1BCHE
SCHEMBL9764389 0.91 ADRB2 (0.39) ADRB2SLC2A1NR1H3ADRB1BCHE
SCHEMBL9764371 0.91 ADRB2 (0.41) ADRB2SLC2A1NR1H3ADRB1BCHE
SCHEMBL9764694 0.89 NR1H3 (0.45) ADRB2NR1H3BCHE
SCHEMBL10346957 0.88 KDM4E (0.40) NR1H3BCHESLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL4950922 0.88 ADRB2 (0.44) ADRB2ADRB1BCHECYP51A1CA12
SCHEMBL10423748 0.88 ADRB2 (0.41) ADRB2NR1H3ADRB1
SCHEMBL9764242 0.87 MC4R (0.39) ADRB2CA12CA1CA2CA4
SCHEMBL9321535 0.86 MAOB (0.37) ADRB2NR1H3ADRB1BCHESLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006556-A Dichloroaniline derivatives for the therapy or prophylaxysis of a disease associated with reversible airway obstruction GLAXO GROUP LIMITED (GB) 1991-04-09 US disclosed
US-4943591-A TREATMENT OF ASTHMA AND BRONCHITIS GLAXO GROUP LIMITED (GB) 1990-07-24 US disclosed
EP-0181709-A1 Dichloroaniline Derivatives GLAXO GROUP LIMITED (GB) 1986-05-21 EP disclosed