SCHEMBL9764242

SCHEMBL9764242

Nc1c(Cl)cc(C(O)CN(CCCCCCOCCc2ccc([N+](=O)[O-])cc2)Cc2ccccc2)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MC4R P32245 1/20 0.39
HRH4 Q9H3N8 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
ADRB2 P07550 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KCNH2 Q12809 3/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HTR2A P28223 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
ACHE P22303 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9764429 0.90 ADRB2 (0.41) ADRB2KCNH2LMNAHTR2A
SCHEMBL9764456 0.90 ADRB2 (0.41) ADRB2KCNH2LMNAHTR2A
SCHEMBL10346971 0.90 MC4R (0.43) MC4RHRH4HRH3KCNH2ALDH1A1
SCHEMBL9764389 0.87 ADRB2 (0.39) ADRB2KCNH2
SCHEMBL9764329 0.87 ADRB2 (0.39) ADRB2CA12CA1CA2CA4
SCHEMBL9764371 0.87 ADRB2 (0.41) ADRB2KCNH2HTR2A
SCHEMBL9764694 0.85 NR1H3 (0.45) ADRB2NPC1KCNH2ALDH1A1
SCHEMBL9764542 0.84 ADRB2 (0.41) ADRB2KCNH2ALDH1A1LMNA
SCHEMBL9764425 0.83 KCNH2 (0.51) ADRB2KCNH2
SCHEMBL9321535 0.82 MAOB (0.37) ADRB2LMNAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006556-A Dichloroaniline derivatives for the therapy or prophylaxysis of a disease associated with reversible airway obstruction GLAXO GROUP LIMITED (GB) 1991-04-09 US disclosed
US-4943591-A TREATMENT OF ASTHMA AND BRONCHITIS GLAXO GROUP LIMITED (GB) 1990-07-24 US disclosed
EP-0181709-A1 Dichloroaniline Derivatives GLAXO GROUP LIMITED (GB) 1986-05-21 EP disclosed