SCHEMBL9764694

SCHEMBL9764694

COc1ccc(CCOCCCCCN(Cc2ccccc2)CC(O)c2cc(Cl)c(N)c(Cl)c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 4/20 0.45
L3MBTL1 Q9Y468 3/20 0.41
TDP1 Q9NUW8 1/20 0.41
MAOB P27338 3/20 0.39
MAOA P21397 1/20 0.39
ADRB2 P07550 1/20 0.38
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
MEP1B Q16820 1/20 0.37
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
BCHE P06276 1/20 0.36
ALOX5 P09917 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9764301 0.96 NR1H3 (0.45) NR1H3L3MBTL1TDP1MAOBMAOA
SCHEMBL9764429 0.93 ADRB2 (0.41) NR1H3MAOBADRB2TSHRBCHE
SCHEMBL9764456 0.93 ADRB2 (0.41) NR1H3MAOBADRB2TSHRBCHE
SCHEMBL9764389 0.91 ADRB2 (0.39) NR1H3ADRB2BCHEKCNH2
SCHEMBL9764329 0.89 ADRB2 (0.39) NR1H3ADRB2BCHE
SCHEMBL9764371 0.89 ADRB2 (0.41) NR1H3ADRB2TSHRBCHEKCNH2
SCHEMBL9324009 0.87 MAOB (0.39) NR1H3MAOBMAOABCHE
SCHEMBL9321535 0.86 MAOB (0.37) NR1H3MAOBMAOAADRB2POLB
SCHEMBL9764542 0.86 ADRB2 (0.41) NR1H3MAOBADRB2ALDH1A1KCNH2
SCHEMBL9764242 0.85 MC4R (0.39) ADRB2NPC1ALDH1A1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006556-A Dichloroaniline derivatives for the therapy or prophylaxysis of a disease associated with reversible airway obstruction GLAXO GROUP LIMITED (GB) 1991-04-09 US disclosed
US-4943591-A TREATMENT OF ASTHMA AND BRONCHITIS GLAXO GROUP LIMITED (GB) 1990-07-24 US disclosed
EP-0181709-A1 Dichloroaniline Derivatives GLAXO GROUP LIMITED (GB) 1986-05-21 EP disclosed