SCHEMBL9764350

SCHEMBL9764350

CC(C)c1c(-c2ccccc2)c(-c2ccc(F)cc2)cn1C(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
HMGCR P04035 4/20 0.42
MEN1 O00255 1/20 0.38
CASP3 P42574 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38
NCOA1 Q15788 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
ALDH1A3 P47895 1/20 0.37
ELAVL1 Q15717 1/20 0.35
ACHE P22303 1/20 0.35
MET P08581 1/20 0.35
CDC25A P30304 1/20 0.34
CDC25C P30307 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9751010 0.78 HMGCR (0.49) KDM4EALDH1A1TDP1L3MBTL1HMGCR
SCHEMBL9518177 0.76 HMGCR (0.47) HMGCR
SCHEMBL9751046 0.75 HMGCR (0.55) ALDH1A1HMGCRMET
SCHEMBL9750967 0.74 HMGCR (0.47) KDM4EHMGCRMEN1KMT2A
SCHEMBL22188201 0.73 KDM4E (0.42) KDM4EALDH1A1TDP1L3MBTL1HMGCR
SCHEMBL6493537 0.73 HMGCR (0.45) HMGCRCYP2C9PTGDRPTGDR2
SCHEMBL10506766 0.72 HMGCR (0.39) HMGCRCDC25ACDC25C
SCHEMBL29941711 0.72 GSK3B (0.48) MEN1KMT2ACDC25ACDC25CCYP2C9
SCHEMBL1878132 0.72 GSK3B (0.48) MEN1KMT2ACDC25ACDC25CCYP2C9
SCHEMBL5731708 0.72 ALDH1A1 (0.50) KDM4EALDH1A1MEN1KMT2ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5032590-A Substituted hydroxylamines BAYER AKTIENGESELLSCHAFT (DE) 1991-07-16 US disclosed
US-4968681-A Substituted hydroxylamines BAYER AKTIENGESELLSCHAFT (DE) 1990-11-06 US disclosed
CN-1033991-A SUBSTITUTED HYDROXYLAMINES BAYER AG (DE) 1989-07-19 CN disclosed
EP-0317845-A2 Substituted hydroxyl amines BAYER AG (DE) 1989-05-31 EP disclosed
EP-0300278-A2 Process for the preparation of 2-substituted pyrroles BAYER AG (DE) 1989-01-25 EP disclosed