SCHEMBL9751046

SCHEMBL9751046

CC(C)c1c(C=O)c(-c2ccc(F)cc2)cn1C(C)C

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 7/20 0.55
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
ALDH1A1 P00352 1/20 0.34
PTGS2 P35354 4/20 0.33
PTGS1 P23219 3/20 0.33
MAPK13 O15264 1/20 0.33
MAPK12 P53778 1/20 0.33
MAPK11 Q15759 1/20 0.33
MAPK14 Q16539 1/20 0.33
MET P08581 1/20 0.33
ERN1 O75460 1/20 0.33
ATM Q13315 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9750945 0.86 HMGCR (0.56) HMGCRADORA2AADORA1PTGS2PTGS1
SCHEMBL9518437 0.86 HMGCR (0.56) HMGCRADORA2AADORA1PTGS2PTGS1
SCHEMBL9750845 0.84 HMGCR (0.56) HMGCRADORA2AADORA1ALDH1A1PTGS2
SCHEMBL9518155 0.81 HMGCR (0.53) HMGCRADORA2AADORA1ALDH1A1MAPK13
SCHEMBL9750837 0.78 HMGCR (0.58) HMGCRALDH1A1PTGS2
SCHEMBL9751010 0.77 HMGCR (0.49) HMGCRADORA2AADORA1ALDH1A1
SCHEMBL9518373 0.76 HMGCR (0.58) HMGCRPTGS2PTGS1MAPK13MAPK12
SCHEMBL9024748 0.75 ELAVL1 (0.45) HMGCRPTGS2PTGS1
SCHEMBL9518177 0.75 HMGCR (0.47) HMGCR
SCHEMBL9764350 0.75 KDM4E (0.43) HMGCRALDH1A1MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5055484-A Anticholesterol and antilipemic agent HOECHST AKTIENGESELLSCHAFT (DE) 1991-10-08 US disclosed