SCHEMBL9764618

SCHEMBL9764618

Oc1c(CN2CCCC2)cc(Cc2ccccc2)cc1CN1CCCC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
HTT P42858 3/20 0.55
HPGD P15428 1/20 0.55
LMNA P02545 3/20 0.52
CYP2D6 P10635 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C19 P33261 1/20 0.50
KDM4E B2RXH2 2/20 0.48
MITF O75030 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
LTA4H P09960 3/20 0.47
ALOX15 P16050 1/20 0.47
ALOX12 P18054 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
PTPN1 P18031 2/20 0.46
PTPN2 P17706 1/20 0.46
PTPN6 P29350 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10011199 0.81 ALDH1A1 (0.56) ALDH1A1HTTLMNACYP2D6CYP2C9
SCHEMBL10008027 0.79 ALDH1A1 (0.59) ALDH1A1HTTCYP2C9CYP3A4KDM4E
SCHEMBL9764604 0.79 HRH3 (0.58) ALDH1A1HTTLMNAKDM4EMITF
SCHEMBL9174306 0.77 PTPN1 (0.70) HPGDCYP3A4ALOX15PTPN1PTPN2
SCHEMBL9804555 0.77 PTPN1 (0.70) HPGDCYP3A4ALOX15PTPN1PTPN2
SCHEMBL29799377 0.76 PRMT6 (0.51) ALDH1A1CYP2D6CYP2C9CYP3A4CYP2C19
SCHEMBL9764649 0.75 LTA4H (0.49) ALDH1A1HPGDLMNACYP2D6CYP2C9
SCHEMBL11209438 0.75 PTPN1 (0.68) HPGDCYP3A4ALOX15PTPN1PTPN2
SCHEMBL30275949 0.75 KDM4E (0.56) ALDH1A1HTTLMNACYP2D6CYP2C9
SCHEMBL9764759 0.75 CACNA1B (0.57) ALDH1A1CYP2D6CYP2C9L3MBTL1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5059620-A Antiarrhythmia agents THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1991-10-22 US disclosed
US-4923873-A ANTIARRHYTHMIA AGENTS; SIDE EFFECT REDUCTION E. I. DU PONT DE NEMOURS AND COMPANY (US) 1990-05-08 US disclosed
US-4755527-A Aryl substituted aminomethyl benzene derivatives E. I. DU PONT DE NEMOURS AND COMPANY (US) 1988-07-05 US disclosed
US-4748184-A Aryl substituted aminomethyl benzene derivatives having antiarrhythmic utility E. I. DU PONT DE NEMOURS AND COMPANY (US) 1988-05-31 US disclosed
US-4562201-A ANTIARRHYTHMIA AGNETS AMERICAN HOSPITAL SUPPLY CORPORATION (US) 1985-12-31 US disclosed
EP-0113778-A4 ARYL SUBSTITUTED AMINOMETHYL BENZENE DERIVATIVES USEFUL AS ANTIARRHYTHMIC AGENTS. AMERICAN HOSPITAL SUPPLY CORP (US) 1985-06-06 EP disclosed
EP-0113778-A1 ARYL SUBSTITUTED AMINOMETHYL BENZENE DERIVATIVES USEFUL AS ANTIARRHYTHMIC AGENTS. AMERICAN HOSPITAL SUPPLY CORP (US) 1984-07-25 EP disclosed
WO-1984000545-A1 ARYL SUBSTITUTED AMINOMETHYL BENZENE DERIVATIVES USEFUL AS ANTIARRHYTHMIC AGENTS AMERICAN HOSPITAL SUPPLY CORP (US) 1984-02-16 WO disclosed