SCHEMBL9765951

SCHEMBL9765951

CC(C)CCn1c(-c2ccccc2)nc2c(=O)[nH]c(=O)n(CC(C)C)c21

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.49
ADORA2B P29275 1/20 0.49
ALDH1A1 P00352 9/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
KDM4E B2RXH2 5/20 0.44
MAPK1 P28482 1/20 0.44
HPGD P15428 4/20 0.44
HSD17B10 Q99714 3/20 0.44
TSHR P16473 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP2C9 P11712 1/20 0.43
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9765921 0.72 ALDH1A1 (0.59) ADORA2AADORA2BALDH1A1SMN1; SMN2KDM4E
SCHEMBL8937183 0.72 KDM4E (0.43) ALDH1A1KDM4EHPGDTSHRMEN1
SCHEMBL23797830 0.71 HTT (0.42) ADORA2AADORA2BALDH1A1KDM4EHSD17B10
SCHEMBL4623478 0.71 KDM4E (0.38) ALDH1A1SMN1; SMN2KDM4EHPGDMEN1
SCHEMBL9765915 0.70 ALDH1A1 (0.52) ADORA2BALDH1A1KDM4EHPGDHSD17B10
SCHEMBL7624092 0.69 KDM4E (0.42) ADORA2AADORA2BALDH1A1SMN1; SMN2KDM4E
SCHEMBL3110932 0.68 PDE1A (0.53) HPGDMEN1KMT2A
SCHEMBL5647 0.67 ADORA2A (0.43) ADORA2AADORA2BALDH1A1KDM4EMAPK1
SCHEMBL1804901 0.67 KDM4E (0.41) ALDH1A1KDM4EHPGDHSD17B10TSHR
SCHEMBL4621732 0.66 ADORA2A (0.43) ADORA2AADORA2BALDH1A1KDM4EMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0383868-A4 1,3-UNSYMMETRICAL STRAIGHT CHAIN ALKYL-SUBSTITUTED 8-PHENYLXANTHINES 1991-12-04 EP disclosed
EP-0383868-A1 1,3-UNSYMMETRICAL STRAIGHT CHAIN ALKYL-SUBSTITUTED 8-PHENYLXANTHINES MARION LABORATORIES, INC. (US) 1990-08-29 EP disclosed
WO-1990000056-A1 1,3-UNSYMMETRICAL STRAIGHT CHAIN ALKYL-SUBSTITUTED 8-PHENYLXANTHINES MARION LABORATORIES, INC. (US) 1990-01-11 WO disclosed