SCHEMBL7624092

SCHEMBL7624092

CC(C)Cn1c(=O)[nH]c(=O)c2nc(Br)n(C)c21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ALDH1A1 P00352 4/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
GAA P10253 2/20 0.39
LMNA P02545 2/20 0.39
PDE1A P54750 3/20 0.38
PDE1B Q01064 3/20 0.38
PDE1C Q14123 3/20 0.38
PDE2A O00408 2/20 0.38
HPGD P15428 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
ADORA3 P0DMS8 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA2B P29275 1/20 0.36
ADORA1 P30542 1/20 0.36
MAPK1 P28482 2/20 0.36
PDE5A O76074 1/20 0.36
TSHR P16473 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8937183 0.84 KDM4E (0.43) KDM4ENPSR1ALDH1A1MEN1KMT2A
SCHEMBL1804901 0.81 KDM4E (0.41) KDM4ENPSR1ALDH1A1MEN1KMT2A
SCHEMBL2476718 0.80 MEN1 (0.45) KDM4ENPSR1ALDH1A1MEN1KMT2A
SCHEMBL19013418 0.78 KDM4E (0.40) KDM4EALDH1A1MEN1KMT2AGAA
SCHEMBL4623478 0.74 KDM4E (0.38) KDM4ENPSR1ALDH1A1MEN1KMT2A
SCHEMBL5647 0.72 ADORA2A (0.43) KDM4ENPSR1ALDH1A1MEN1KMT2A
SCHEMBL9765951 0.69 ADORA2A (0.49) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL4796600 0.69 PDE4A (0.47) KDM4EALDH1A1MEN1KMT2AGAA
SCHEMBL23797830 0.69 HTT (0.42) KDM4EALDH1A1MEN1KMT2AGAA
SCHEMBL4623658 0.68 PDE4A (0.39) KDM4ENPSR1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1208100-A1 SELECTIVE ANTAGONISTS OF A2B ADENOSINE RECEPTORS VANDERBILT UNIVERSITY (US) 2002-05-29 EP disclosed
WO-2001016134-A1 SELECTIVE ANTAGONISTS OF A2B ADENOSINE RECEPTORS VANDERBILT UNIVERSITY (US) 2001-03-08 WO disclosed