SCHEMBL9766005

SCHEMBL9766005

O=C(CCN1CCN(c2ncc(F)cn2)CC1)Cc1cccs1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.50
SIGMAR1 Q99720 6/20 0.46
DRD2 P14416 2/20 0.46
KDM4E B2RXH2 1/20 0.46
CYP1A2 P05177 1/20 0.46
GAA P10253 1/20 0.46
CYP2C9 P11712 1/20 0.46
ADRA2C P18825 1/20 0.45
DRD4 P21917 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HRH1 P35367 1/20 0.45
DRD3 P35462 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9766013 0.80 SIGMAR1 (0.60) HTR1ASIGMAR1DRD2KDM4ECYP1A2
SCHEMBL9199690 0.79 HTT (0.56) GAA
SCHEMBL9120369 0.79 KMT2A (0.60) SIGMAR1CYP1A2GAACYP2C9
SCHEMBL9766014 0.79 HTR1A (0.57) HTR1ASIGMAR1DRD2KDM4ECYP1A2
Hydrochloric Acid SCHEMBL9119984 0.78 ALDH1A1 (0.56) GAA
SCHEMBL9207862 0.78 KMT2A (0.58) SIGMAR1CYP1A2GAACYP2C9
SCHEMBL9121156 0.78 KMT2A (0.58) SIGMAR1CYP1A2GAACYP2C9
Hydrochloric Acid SCHEMBL9122307 0.78 KMT2A (0.58) SIGMAR1GAA
SCHEMBL9766069 0.77 SIGMAR1 (0.67) HTR1ASIGMAR1DRD2KDM4ECYP1A2
Hydrochloric Acid SCHEMBL9120318 0.76 KMT2A (0.57) SIGMAR1CYP1A2GAACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0400661-A1 Agents for treatment of brain ischemia Bristol-Myers Squibb Company (US) 1990-12-05 EP claimed
US-4994460-A Treatment or prevention of disorders resulting from central nervous system anoxia BRISTOL-MYERS SQUIBB CO. (US) 1991-02-19 US disclosed
EP-0400661-A1 Agents for treatment of brain ischemia Bristol-Myers Squibb Company (US) 1990-12-05 EP disclosed