SCHEMBL9767412

SCHEMBL9767412

CCC1Oc2ccc(C#N)cc2C2OC12

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.38
DRD3 P35462 4/20 0.38
ABCB1 P08183 10/20 0.36
KCNE1 P15382 4/20 0.36
KCNQ1 P51787 4/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
KCND3 Q9UK17 1/20 0.36
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9767096 0.87 DRD2 (0.38) DRD2DRD3ABCB1KCNE1KCNQ1
SCHEMBL9767595 0.81 ABCB1 (0.39) DRD2DRD3ABCB1KDM4E
SCHEMBL9767236 0.75 KCNE1 (0.40) DRD2DRD3ABCB1KCNE1KCNQ1
SCHEMBL9767232 0.75 KCNE1 (0.40) DRD2DRD3ABCB1KCNE1KCNQ1
SCHEMBL9765458 0.68 ABCB1 (0.43) ABCB1KCNE1KCNQ1MEN1CYP1A2
SCHEMBL13594010 0.67 ABCB1 (0.42) DRD2DRD3ABCB1KCNE1KCNQ1
SCHEMBL9767316 0.67 ABCB1 (0.46) ABCB1KCNE1KCNQ1MEN1CYP1A2
SCHEMBL9766986 0.66 KCNE1 (0.41) DRD2DRD3ABCB1KCNE1KCNQ1
SCHEMBL9766987 0.66 KCNE1 (0.41) DRD2DRD3ABCB1KCNE1KCNQ1
SCHEMBL482249 0.65 ABCB1 (0.56) ABCB1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5072006-A Chemical intermeidate; hypotensive agents, muscle relaxants RECHERCHE SYNTEX FRANCE S.A. (FR) 1991-12-10 US disclosed
US-4997846-A Smooth muscle relaxants, hypotensives RESEARCHE SYNTEX FRANCE, S.A. (FR) 1991-03-05 US disclosed
EP-0377966-A2 Novel benzopyranylpyrrolinone derivatives RECHERCHE SYNTEX FRANCE SA (FR) 1990-07-18 EP disclosed