SCHEMBL9767565

SCHEMBL9767565

CCCNc1ccncc1N1CCCc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
KMT2A Q03164 1/20 0.42
KDM4C Q9H3R0 5/20 0.42
ROCK1 Q13464 1/20 0.41
NUDT1 P36639 1/20 0.40
KDM6B O15054 2/20 0.39
POLB P06746 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
AVPR2 P30518 1/20 0.38
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37
TUBB3 Q13509 1/20 0.37
TUBB2A Q13885 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9195257 0.78 ROCK1 (0.52) MEN1ALDH1A1KMT2AKDM4CROCK1
Hydrochloric Acid SCHEMBL9767541 0.77 ROCK1 (0.51) MEN1ALDH1A1KMT2AKDM4CROCK1
SCHEMBL9196015 0.72 ALDH1A1 (0.52) MEN1ALDH1A1KMT2AKDM4CPOLB
SCHEMBL9193973 0.69 ROCK1 (0.50) MEN1ALDH1A1KMT2AROCK1POLB
SCHEMBL9192032 0.69 EED (0.52) MEN1ALDH1A1KMT2AROCK1POLB
SCHEMBL1102659 0.69 ROCK1 (0.48) ALDH1A1KMT2AKDM4CROCK1NUDT1
SCHEMBL26103577 0.68 SMN1; SMN2 (0.48) MEN1ALDH1A1KMT2AROCK1POLB
SCHEMBL9767604 0.68 ALOX15 (0.51) MEN1ALDH1A1KMT2AKDM4CROCK1
Maleic Acid SCHEMBL9767806 0.67 ALDH1A1 (0.46) ALDH1A1KDM4CKDM6BPOLBL3MBTL1
Fumaric Acid SCHEMBL9767822 0.67 ALDH1A1 (0.46) ALDH1A1KDM4CKDM6BPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4992448-A Benzocycloalkylaminopyridinamines and related compounds as topical antiinflammatory agents for the treatment of skin disorders HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-02-12 US claimed
US-5037835-A Benzocycloalkylaminopyridinamines and related compounds as topical antiinflammatory agents for the treatment of skin disorders HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-08-06 US disclosed
EP-0428878-A2 Benzocycloalkylaminopyridinamines and related compounds, a process and intermediates for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-05-29 EP disclosed
US-4992448-A Benzocycloalkylaminopyridinamines and related compounds as topical antiinflammatory agents for the treatment of skin disorders HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-02-12 US disclosed