SCHEMBL9768785

SCHEMBL9768785

CN1c2ccccc2N(C(=O)CCl)c2ccccc2S1(=O)=O

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.53
MITF O75030 1/20 0.53
RAB9A P51151 1/20 0.53
ALDH1A1 P00352 2/20 0.39
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
TP53 P04637 1/20 0.38
CASP3 P42574 1/20 0.37
CASP2 P42575 1/20 0.37
NR1I2 O75469 2/20 0.36
HSD11B1 P28845 1/20 0.36
OPRM1 P35372 1/20 0.36
DRD3 P35462 1/20 0.36
OPRD1 P41143 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9768762 0.89 NPC1 (0.40) NPC1MITFRAB9AALDH1A1CA2
SCHEMBL9768766 0.88 NPC1 (0.45) NPC1MITFRAB9AALDH1A1TP53
SCHEMBL9768711 0.88 NPC1 (0.45) NPC1MITFRAB9AALDH1A1NR1I2
SCHEMBL9768779 0.88 NPC1 (0.45) NPC1MITFRAB9AALDH1A1NR1I2
SCHEMBL9768790 0.87 NPC1 (0.46) NPC1MITFRAB9AALDH1A1NR1I2
SCHEMBL9768718 0.87 NR1I2 (0.46) NPC1MITFRAB9AALDH1A1CA2
SCHEMBL9768904 0.84 CYP1A2 (0.48) NPC1MITFRAB9AALDH1A1CYP1A2
SCHEMBL9768684 0.83 ALDH1A1 (0.50) NPC1MITFRAB9AALDH1A1CA9
SCHEMBL9768760 0.83 KDM4E (0.48) NPC1MITFRAB9AALDH1A1CA2
SCHEMBL9768832 0.83 MTNR1A (0.40) CA2CA9TP53HSD11B1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5011833-A Antidepressant A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE (IT) 1991-04-30 US disclosed
EP-0354885-A1 Novel derivatives of 6,11-dihydro-dibenzo[c,f][1,2,5]-thiadiazepine 5,5-dioxide, salts thereof and appropriate processes for the preparation thereof A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1990-02-14 EP disclosed